A cross-species translational pharmacokinetic-pharmacodynamic evaluation of core body temperature reduction by the TRPM8 blocker PF-05105679

Therapeutic area :

Gosset J.R., Beaumont K., Matsuura T., Winchester W., Attkins N., Glatt S.,Lightbown I., Ulrich K., Roberts S., Harris J., Mesic E., Steeg T.J.v., Hijdra D., Graaf P.H.v.d.  A cross-species translational pharmacokinetic-pharmacodynamic evaluation of core body temperature reduction by the TRPM8 blocker PF-05105679. European Journal of Pharmaceutical Sciences: S161-S167 2017. [Link to publication]