Publications

A model-based approach to analyze the influence of UGT2B15

Stringer F., Dejongh J., Scott G. and Danhof M., A model-based approach to analyze the influence of UGT2B15 polymorphism driven pharmacokinetic differences on the pharmacodynamic response of the PPAR agonist sipoglitazar, J Clin Pharmacol, 11(10): 227, 2013. [Link to publication]

Pharmacokinetics of Recombinant Human Antithrombin

Dejongh J., Frieling J., Lowry S. and Drenth H.J., Pharmacokinetics of Recombinant Human Antithrombin in Delivery and Surgery Patients With Hereditary Antithrombin Deficiency, Clin Appl Thromb Hemost, 11: 11, 2013. [Link to publication]

Application of M&S for Bispecifics in early discorvery.

Steeg T.v., Bergmann K., agoram B. and Sachsenmeier K., Application of M&S for Bispecifics in early discorvery. PKPK of novel constructs.(2013)

Acute dopamine inhibition challenge

Stevens J., Ploeger B.A., Hammarlund-Udenaes M., Osswald G., van der Graaf P.H., Danhof M. and de Lange E.C., Mechanism-based PK-PD model for the prolactin biological system response following an acute dopamine inhibition challenge: quantitative extrapolation to humans, J Pharmacokinet Pharmacodyn., 39(5): 463-477. 2012. [Link to publication]

Regional brain distribution kinetics in rats

Westerhout J., Ploeger B., Smeets J., Danhof M. and de Lange E.C., Physiologically based pharmacokinetic modeling to investigate regional brain distribution kinetics in rats, Aaps J., 14(3): 543-553. doi: 510.1208/s12248-12012-19366-12241. Epub 12012 May 12217., 2012. [Link to publication]

Evaluation of blood-brain barrier transport and CNS drug metabolism

Ravenstijn P.G., Drenth H.J., O’Neill M.J., Danhof M. and de Lange E.C., Evaluation of blood-brain barrier transport and CNS drug metabolism in diseased and control brain after intravenous L-DOPA in a unilateral rat model of Parkinson’s disease, Fluids Barriers CNS., 9:4. 2012. [Link to publication]

Drug-induced sleep fragmentation

Diack C., Ackaert O., Ploeger B.A., Graaf  P.H.v.d., Gurrell R., Ivarsson M., and Fairman D. A hidden Markov model to assess drug-induced sleep fragmentation in the telemetered rat, J Pharmacokinet Pharmacodyn, 10: 10, 2011. [Link to publication]

Morphine and its metabolites

Krekels E.H., Jongh J.d., Lingen R.A.v., Marel C.D.v.d., Choonara I., Lynn A.M., Danhof M., Tibboel D. and Knibbe C.A., Predictive performance of a recently developed population pharmacokinetic model for morphine and its metabolites in new datasets of (preterm) neonates, infants and children, Clin Pharmacokinet., 50(1): 51-63, 2011. [Link to publication]

Predictive performance in simulation models of clinical trials

Holford N., Ma S.C. and Ploeger B.A., Response to “validation and assessment of predictive performance in simulation models of clinical trials”, Clin Pharmacol Ther., 89(4): 488. 2011. [Link to publication]

Effect on CYP3A4 activity

Erp N.P.v., Guchelaar H.J., Ploeger B.A., Romijn J.A., Hartigh J. and Gelderblom H., Mitotane has a strong and a durable inducing effect on CYP3A4 activity, Eur J Endocrinol., 164(4): 621-626. 2011. [Link to publication]