Publications

Pharmacokinetic-pharmacodynamic modelling of fluvoxamine 5-HT transporter occupancy in rat frontal cortex

Geldof M., Freijer J.I., Beijsterveldt L.v., Langlois X. and Danhof M., Pharmacokinetic-pharmacodynamic modelling of fluvoxamine 5-HT transporter occupancy in rat frontal cortex, Br J Pharmacol., 154(6): 1369-1378. Epub 2008 May 1319., 2008.  [Link to publication]

Mechanistic model for the acute effect of fluvoxamine on 5-HT and 5-HIAA concentrations

Geldof M., Freijer J.I., Peletier L.A., Beijsterveldt L.v. and Danhof M., Mechanistic model for the acute effect of fluvoxamine on 5-HT and 5-HIAA concentrations in rat frontal cortex, Eur J Pharm Sci., 33(3): 217-229. Epub 2007 Dec 2007., 2008. [Link to publication]

Pharmacokinetic modeling of non-linear brain distribution of fluvoxamine in the rat

Geldof M., Freijer J., Beijsterveldt L.v. and Danhof M., Pharmacokinetic modeling of non-linear brain distribution of fluvoxamine in the rat, Pharm Res., 25(4): 792-804. Epub 2007 Aug 2021., 2008. [Link to publication]

Amoxicillin pharmacokinetics in pregnant women

Muller A.E., Jongh J.d., Oostvogel P.M., Voskuyl R.A., Dorr P.J., Danhof M. and Mouton J.W., Amoxicillin pharmacokinetics in pregnant women with preterm premature rupture of the membranes, Am J Obstet Gynecol, 198(1): 108 e101-106, 2008. [Link to publication]

Mechanism-based pharmacodynamic modeling of S(-)-atenolol

Steeg T.J.v., Freijer J., Danhof M.  and Lange E. C. d., Mechanism-based pharmacodynamic modeling of S(-)-atenolol: estimation of in vivo affinity for the beta1-adrenoceptor with an agonist-antagonist interaction model, J Pharmacol Exp Ther., 324(3): 1234-1242., 2008. [Link to publication]

The influence of labour on the pharmacokinetics of intravenously administered amoxicillin in pregnant women

Muller A.E., Dorr P.J., Mouton J.W., Jongh J.d., Oostvogel P.M., Steegers E.A., Voskuyl R.A. and Danhof M., The influence of labour on the pharmacokinetics of intravenously administered amoxicillin in pregnant women, Br J Clin Pharmacol., 66(6): 866-874., 2008. [Link to publication]

Extensions to the visual predictive check to facilitate model performance evaluation,

Post T.M., Freijer J.I., Ploeger B.A. and Danhof M., Extensions to the visual predictive check to facilitate model performance evaluation, J Pharmacokinet Pharmacodyn., 35(2): 185-202. 2008. [Link to publication]

Mechanism-based pharmacokinetic-pharmacodynamic (PK-PD) modeling

Danhof M., Lange E.C.d, Della Pasqua O.E., Ploeger B.A. and Voskuyl R.A., Mechanism-based pharmacokinetic-pharmacodynamic (PK-PD) modeling in translational drug research, Trends Pharmacol Sci., 29(4): 186-191., 2008. [Link to publication]

Pharmacokinetic/pharmacodynamic modelling of the EEG effects of opioids

Groenendaal D., Freijer J., Rosier A., Mik D.d., Nicholls G., Hersey A., Ayrton A.D., Danhof M. and Lange E.C.d., Pharmacokinetic/pharmacodynamic modelling of the EEG effects of opioids: the role of complex biophase distribution kinetics, Eur J Pharm Sci., 34(2-3): 149-163. Epub 2008 Mar 2030., 2008. [Link to publication]

Pharmacokinetic-pharmacodynamic modelling of S(-)-atenolol in rats

Steeg T.J.v., Freijer J., Danhof M. and Lange E.C.d, Pharmacokinetic-pharmacodynamic modelling of S(-)-atenolol in rats: reduction of isoprenaline-induced tachycardia as a continuous pharmacodynamic endpoint, Br J Pharmacol, 10: 10, 2007. [Link to publication]